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Busulfan, Fludarabine Phosphate, and Anti-Thymocyte Globulin Followed By Donor Stem Cell Transplant and Azacitidine in Treating Patients With High-Risk Myelodysplastic Syndrome and Older Patients With Acute Myeloid Leukemia

Phase II Study of the Addition of Azacitidine (NSC#102816) to Reduced-Intensity Conditioning Allogeneic Transplantation for Myelodysplasia (MDS) and Older Patients With AML

Status
Completed
Phases
Phase 2
Study type
Interventional
Source
ClinicalTrials.gov
Registry ID
NCT01168219
Enrollment
68
Registered
2010-07-23
Start date
2010-07-15
Completion date
2020-02-01
Last updated
2022-08-04

For informational purposes only — not medical advice. Sourced from public registries and may not reflect the latest updates. Terms

Conditions

Acute Myeloid Leukemia, Adult Acute Megakaryoblastic Leukemia, Adult Acute Monoblastic Leukemia, Adult Acute Monocytic Leukemia, Adult Acute Myeloid Leukemia With Inv(16)(p13.1q22); CBFB-MYH11, Adult Acute Myeloid Leukemia With Maturation, Adult Acute Myeloid Leukemia With Minimal Differentiation, Adult Acute Myeloid Leukemia Without Maturation, Adult Acute Myeloid Leukemia With t(16;16)(p13.1;q22); CBFB-MYH11, Adult Acute Myeloid Leukemia With t(8;21); (q22; q22.1); RUNX1-RUNX1T1, Adult Acute Myeloid Leukemia With t(9;11)(p21.3;q23.3); MLLT3-MLL, Adult Acute Myelomonocytic Leukemia, Adult Erythroleukemia, Adult Pure Erythroid Leukemia, Alkylating Agent-Related Acute Myeloid Leukemia, de Novo Myelodysplastic Syndrome, Myelodysplastic Syndrome, Myelodysplastic Syndrome With Excess Blasts, Recurrent Adult Acute Myeloid Leukemia, Secondary Myelodysplastic Syndrome

Brief summary

This phase II clinical trial is studying how well giving busulfan, fludarabine phosphate, and anti-thymocyte globulin followed by donor stem cell transplant and azacitidine works in treating patients with high-risk myelodysplastic syndrome and older patients with acute myeloid leukemia. Giving low doses of chemotherapy, such as busulfan and fludarabine phosphate, before a donor stem cell transplant helps stop the growth of cancer cells. It also stops the patient's immune system from rejecting the donor's stem cells. The donated stem cells may replace the patient's immune cells and help destroy any remaining cancer cells (graft-vs-tumor effect). Sometimes the transplanted cells from a donor can also make an immune response against the body's normal cells. Giving anti-thymocyte globulin before transplant and giving azacitidine, tacrolimus, and methotrexate after the transplant may stop this from happening.

Detailed description

PRIMARY OBJECTIVE: I. To determine if this treatment can improve 2-year progression-free survival (PFS) in patients with high risk myelodysplastic syndrome (MDS) and in patients with acute myeloid leukemia (AML) \>= 60 yrs age SECONDARY OBJECTIVES: I. To determine the safety and feasibility of using post-transplantation azacitidine. II. To determine the ability to use pharmacokinetic-directed busulfan to achieve area under the curve (AUC) within 20% of target AUC in \> 80% of patients. III. To determine the rate of grade II-IV and III-IV acute graft-vs-host disease (GVHD). IV. To determine the incidence of extensive chronic GVHD. V. To determine treatment-related mortality at 100 days and at 1 year. VI. To determine 5-year overall survival. OUTLINE: REDUCED-INTENSITY CONDITIONING: Patients receive fludarabine phosphate intravenously (IV) over 30 minutes on days -7 to -3, busulfan IV over 45 minutes on days -6 to -3, and anti-thymocyte globulin IV over 4-10 hours on days -6 to -5 (matched sibling donor \[MSD\]) or -6 to -4 (matched unrelated donor \[MUD\]). TRANSPLANTATION: Patients undergo allogeneic hematopoietic stem cell transplantation on day 0 or on days 0-1. GRAFT-VS-HOST DISEASE PROPHYLAXIS: Patients receive tacrolimus orally (PO) or IV on days -2 to 90 with taper on days 150-180. Patients also receive methotrexate IV on days 1, 3, 6 (MSD), and 11 (MUD). CONSOLIDATION: Beginning on day 42, patients receive azacitidine subcutaneously (SC) or IV on days 1-5. Treatment repeats every 4 weeks for 6 courses. Blood and bone marrow samples may be collected periodically for correlative and pharmacokinetic studies. After completion of study treatment, patients are followed up every 6 months for 5 years.

Interventions

PROCEDUREAllogeneic Hematopoietic Stem Cell Transplantation

Undergo allogeneic hematopoietic stem cell transplantation

BIOLOGICALAnti-Thymocyte Globulin

Given IV

DRUGAzacitidine

Given SC or IV

DRUGBusulfan

Given IV

DRUGFludarabine Phosphate

Given IV

OTHERLaboratory Biomarker Analysis

Correlative studies

DRUGMethotrexate

Given IV

OTHERPharmacological Study

Correlative studies

DRUGTacrolimus

Given PO or IV

Sponsors

National Cancer Institute (NCI)
Lead SponsorNIH

Study design

Allocation
NA
Intervention model
SINGLE_GROUP
Primary purpose
TREATMENT
Masking
NONE

Eligibility

Sex/Gender
ALL
Age
18 Years to 74 Years
Healthy volunteers
No

Inclusion criteria

* Meets one of the following sets of criteria: * Myelodysplastic syndromes (MDS): * Disease with high-risk features (found either at diagnosis or before initiation of cytotoxic therapy), defined as one of the following: * International prognostic scoring system (IPSS) risk \>= intermediate-2 * Refractory anemia with excess blasts by French-American-British (FAB) classification * High-risk cytogenetics (either complex or -7) * Less than 10% bone marrow blasts as determined by bone marrow biopsy within the past 4 weeks (reduction in marrow blast percentage may be achieved with chemotherapy or other therapy) * Less than 75 years old * Acute myeloid leukemia (AML): * No FAB M3 * No acute leukemia following blast transformation of prior chronic myelogenous leukemia or other myeloproliferative disease * Patients with preceding MDS or treatment-related AML are eligible * Prior central nervous system (CNS) involvement is allowed provided the disease is in remission at transplantation * Morphologic complete remission (leukemia-free state) is defined as meeting all of the following criteria: * Bone marrow blasts \< 5% (as determined by bone marrow within the past 4 weeks), but without requirement for normal peripheral blood counts * No extramedullary leukemia * No blasts in peripheral blood * Achieved complete remission (CR) after no more than 2 courses of induction chemotherapy * Patients treated with azacitidine or decitabine who achieve a leukemia-free state are eligible (may have required up to 4 courses of therapy to reach this status) * Age 60 to 74 years * Donors must meet the following criteria: * One of the following: * HLA-identical sibling (6/6) by serologic typing for class (A, B) and low-resolution molecular typing for class II (DRB1) * Matched unrelated donor (8/8) by high-resolution molecular typing at HLA-A, -B, -C, and DRB1 * No syngeneic donors * Eastern Cooperative Oncology Group (ECOG) performance status 0-2 * Calculated creatinine clearance ≥ 40 mL/min * Bilirubin \< 2 mg/dL OR bilirubin 2-3 mg/dL provided direct bilirubin is normal * Aspartate aminotransferase (AST) \< 3 times upper limit of normal * Diffusing capacity of the lung for carbon monoxide (DLCO) \> 40% with no symptomatic pulmonary disease * Left ventricle ejection fraction (LVEF) \>= 30% by echocardiogram (ECHO) or multigated acquisition (MUGA) * Not pregnant or nursing * Negative pregnancy test * Fertile patients must use effective contraception * No uncontrolled diabetes mellitus or active serious infections * No known hypersensitivity to E. coli-derived products, azacitidine, or mannitol * No human immunodeficiency virus (HIV) infection or active hepatitis B or C * Prior azacitidine or decitabine allowed * No patients who progressed from MDS to AML during treatment with azacitidine or decitabine * At least 4 weeks since prior deoxyribonucleic acid (DNA)-hypomethylating chemotherapy, radiotherapy, and/or surgery * No more than 2 courses of consolidation therapy before transplantation (for patients with AML) * Any consolidation regimen that does not require transplantation can be used * No more than 6 months from documentation of morphologic CR to transplantation

Design outcomes

Primary

MeasureTime frameDescription
Progression-free SurvivalUp to 5 yearsProgression-free survival rate (percentage) at 2 and 5 years is defined as the percentage of patients who are alive and progression free at 2 and 5 years from date of transplantation respectively. AML progression is defined as: * Reappearance of leukemia blast cells in peripheral blood and \> 5% blasts in marrow * If no circulating blasts, but the marrow contains 5-20% blasts, a repeat bone marrow \>= 1 week later with \> 5% blasts * Development of extramedullary leukemia MDS progression is defined as * For patients with \<5% bone marrow blasts: ≥50% increase in blasts to \>5% blasts * For patients with 5-10% bone marrow blasts: ≥50% increase to \>10% blasts * Any of the following: Reappearance of prior documented characteristic cytogenetic abnormality or refractory cytopenias with unequivocal evidence of dysplasia on bone marrow biopsy/aspirate

Secondary

MeasureTime frameDescription
100-day MortalityUp to 100 days post-treatmentThe number of death reported within the first 100 days after transplant.
Overall Survival (OS)Up to 5 yearsOverall survival rate (percentage) at 2 and 5 years is defined as the percentage of patients who are still alive 2 and 5 years after date of transplantation respectively. Estimated using the Kaplan-Meier product limit estimator.

Countries

United States

Participant flow

Recruitment details

From July 2010 and October 2013, a total of 68 participants were recruited to this study.

Participants by arm

ArmCount
Treatment (Chemotherapy and Transplant)
REDUCED-INTENSITY CONDITIONING: Patients receive fludarabine phosphate IV over 30 minutes on days -7 to -3, busulfan IV over 45 minutes on days -6 to -3, and anti-thymocyte globulin IV over 4-10 hours on days -6 to -5 (matched sibling donor \[MSD\]) or -6 to -4 (matched unrelated donor \[MUD\]). TRANSPLANTATION: Patients undergo allogeneic hematopoietic stem cell transplantation on day 0 or on days 0-1. GRAFT-VS-HOST DISEASE PROPHYLAXIS: Patients receive tacrolimus PO or IV on days -2 to 90 with taper on days 150-180. Patients also receive methotrexate IV on days 1, 3, 6 (MSD), and 11 (MUD). CONSOLIDATION: Beginning on day 42, patients receive azacitidine SC or IV on days 1.
68
Total68

Withdrawals & dropouts

PeriodReasonFG000
Overall Studyineligible due to CML2
Overall Studyoff study before starting treatment2
Overall Studywithdrew before transplant1

Baseline characteristics

CharacteristicTreatment (Chemotherapy and Transplant)
Age, Continuous62.9 years
Disease type
Acute Myeloid Leukemia (AML)
44 Participants
Disease type
Myelodysplastic Syndrome (MDS)
24 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
3 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
61 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
4 Participants
Race (NIH/OMB)
American Indian or Alaska Native
1 Participants
Race (NIH/OMB)
Asian
2 Participants
Race (NIH/OMB)
Black or African American
1 Participants
Race (NIH/OMB)
More than one race
2 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
Race (NIH/OMB)
Unknown or Not Reported
2 Participants
Race (NIH/OMB)
White
60 Participants
Region of Enrollment
United States
68 Participants
Sex: Female, Male
Female
15 Participants
Sex: Female, Male
Male
53 Participants

Adverse events

Event typeEG000
affected / at risk
deaths
Total, all-cause mortality
42 / 66
other
Total, other adverse events
61 / 66
serious
Total, serious adverse events
22 / 66

Outcome results

Primary

Progression-free Survival

Progression-free survival rate (percentage) at 2 and 5 years is defined as the percentage of patients who are alive and progression free at 2 and 5 years from date of transplantation respectively. AML progression is defined as: * Reappearance of leukemia blast cells in peripheral blood and \> 5% blasts in marrow * If no circulating blasts, but the marrow contains 5-20% blasts, a repeat bone marrow \>= 1 week later with \> 5% blasts * Development of extramedullary leukemia MDS progression is defined as * For patients with \<5% bone marrow blasts: ≥50% increase in blasts to \>5% blasts * For patients with 5-10% bone marrow blasts: ≥50% increase to \>10% blasts * Any of the following: Reappearance of prior documented characteristic cytogenetic abnormality or refractory cytopenias with unequivocal evidence of dysplasia on bone marrow biopsy/aspirate

Time frame: Up to 5 years

Population: Patients who received transplant were evaluable for the primary endpoint.

ArmMeasureGroupValue (NUMBER)
Treatment (Chemotherapy and Transplant)Progression-free SurvivalPFS at 2 years41.2 percentage of patients
Treatment (Chemotherapy and Transplant)Progression-free SurvivalPFS at 5 years26.9 percentage of patients
Secondary

100-day Mortality

The number of death reported within the first 100 days after transplant.

Time frame: Up to 100 days post-treatment

Population: Patients who received transplant and died are included in this analysis.

ArmMeasureValue (COUNT_OF_PARTICIPANTS)
Treatment (Chemotherapy and Transplant)100-day Mortality10 Participants
Secondary

Overall Survival (OS)

Overall survival rate (percentage) at 2 and 5 years is defined as the percentage of patients who are still alive 2 and 5 years after date of transplantation respectively. Estimated using the Kaplan-Meier product limit estimator.

Time frame: Up to 5 years

Population: Patients who received transplant were evaluable for this endpoint.

ArmMeasureGroupValue (NUMBER)
Treatment (Chemotherapy and Transplant)Overall Survival (OS)OS at 2 years45.7 percentage of patients
Treatment (Chemotherapy and Transplant)Overall Survival (OS)OS at 5 years31.2 percentage of patients

Source: ClinicalTrials.gov · Data processed: Mar 2, 2026